Protease Inhibitors and Phosphatase Inhibitors
Echelon Biosciences Research Labs SS14 Tumor Inhibitor Analog - 1 mg,
SS14 Tumor Inhibitor Analog - 1mg , D-Nal-Cys-Tyr-D-Trp-Lys-Val-Cys-Thr-NH2 Category/Application: Neuropeptides Hormones This item is non returnable
Enzo Life Sciences Cystatin C (human), (purified) (100 µg)
Alternative name: Cystatin 3, Neuroendocrine basic polypeptide, CysC. Purity: ≥95% (SDS-PAGE). Formulation: Lyophilized from 0.02M ammonium bicarbonate buffer. Source: Isolated from human urine. Long Term Storage: -20°C.
Echelon Biosciences Research Labs SS14 Tumor Inhibitor Analog - 5 mg,
SS14 Tumor Inhibitor Analog - 5mg , D-Nal-Cys-Tyr-D-Trp-Lys-Val-Cys-Thr-NH2 Category/Application: Neuropeptides Hormones This item is non returnable
Echelon Biosciences Research Labs Caspase 8 Substrate - 5 mg,
Caspase 8 Substrate - 0.5mg , Ac-Val-Glu-Thr-Asp-AMC Category/Application: Enzyme Substrates This item is non returnable
Echelon Biosciences Research Labs MMP-3 Inhibitor 1 - 1 mg,
MMP-3 Inhibitor 1 - 1mg , Ac-Arg-Cys-Gly-Val-Pro-Asp-NH2 Category/Application: Enzyme Substrates This item is non returnable
Cayman Chemical PRL-3 InhIbItr 10mg
A cell-permeable benzylidene rhodamine that inhibits PRL-3 (IC50 = 900 nM for human PRL-3 in vitro), with minimal activity against other phosphatases; reduces the invasion of mouse melanoma B16F10 cells in a cell-based assay
Cayman Chemical K-Ras G12C InhIbItr 9 5mg
An irreversible, allosteric inhibitor of the K-Ras(G12C) mutant that causes 100% modification of the protein when used at 10 µM for 24 hours in vitro
CPC Scientific MCA-Pro-Cha-Gly-Nva-His-Ala-Dap(DNP)-NH2 (trifluoroacetate salt) 0.5MG
Specific fluorogenic substrate for collagenase-3 (MMP) with a kcat/Km value of 1.09 x 106 M-1s-1 (pH = 7.5, T = 25 °C, substrate concentrations: 0.7 and 1.4 µM (S<
Cayman Chemical Cdk2 InhIbItr II 500ug
A 3-(benzylidne)indolin-2-one analog that selectively and potently inhibits Cdk2 (IC50 = 60 nM)
Cayman Chemical PD-1PD-L1 InhIbItr 1 25mg
A PD-1/PD-L1 interaction inhibitor; inhibits the PD-1/PD-L1 interaction in a TR-FRET assay (IC50 = 6-100 nM); reduces LPS-induced increases in PD-1 levels and apoptosis in MH-S mouse alveolar macrophages at 1 µM; surgical neointimal patching with PD-1/PD-L1-coated patches decreases neointimal thickness and inflammatory cell accumulation in a rat model of patch angioplasty
Cayman Chemical FTase InhIbItr IItrIfluoro 5mg
A cell-permeable analog of FPP that potently inhibits FTase (IC50 = 50-75 nM), preventing farnesylation of Ras; does not inhibit geranylgeranyl transferase at similar concentrations (IC50 > 100 µM); blocks Ras-mediated transformation of NIH 3T3 cells